Drug Targeting

Mycobacterium tuberculosis interactome analysis unravels potential pathways to drug resistance

Drug Discovery / Biological Sciences / Tuberculosis / Mycobacterium tuberculosis / Drug Resistance / Shortest Path / Drug Targeting / Drug treatment / Shortest Path / Drug Targeting / Drug treatment

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Pharmacology / Neuroscience / Immunology / Molecular Medicine / Treatment / Drug Discovery / Biological Sciences / Humans / Cholesterol / Vaccination / Metabolic pathway / Brain Chemistry / Drug Targeting / Alzheimer Disease / Drug Discovery / Biological Sciences / Humans / Cholesterol / Vaccination / Metabolic pathway / Brain Chemistry / Drug Targeting / Alzheimer Disease

The intracellular uptake of CD95 modified paclitaxel-loaded poly(lactic-co-glycolic acid) microparticles

Biomaterials / Cancer / Flow Cytometry / Drug delivery / Ovarian Cancer / Multidisciplinary / Humans / Surface modification / Paclitaxel / CD / Immune Evasion / Phagocytosis / Microspheres / Drug Targeting / Drug Carriers / Lactic Acid / Multidisciplinary / Humans / Surface modification / Paclitaxel / CD / Immune Evasion / Phagocytosis / Microspheres / Drug Targeting / Drug Carriers / Lactic Acid

Transport processes in Plasmodium falciparum-infected erythrocytes: potential as new drug targets

Microbiology / Zoology / Transport Properties / Animals / Host-parasite interactions / Membrane transport proteins / Substrate Specificity / Plasmodium falciparum / For / Veterinary Sciences / Heterologous Expression / Erythrocytes / Drug Targeting / Plasma Membrane / Membrane transport proteins / Substrate Specificity / Plasmodium falciparum / For / Veterinary Sciences / Heterologous Expression / Erythrocytes / Drug Targeting / Plasma Membrane

Entamoeba histolytica: Biochemical characterization of a protein disulfide isomerase

Microbiology / Protein Folding / Life Style / Molecular chaperones / Experimental parasitology / Insulin / Oxidoreductases / Enzyme / Experimental / Anti-Bacterial Agents / Entamoeba histolytica / Veterinary Sciences / Drug Targeting / Hydrogen-Ion Concentration / Disulfide bond / Insulin / Oxidoreductases / Enzyme / Experimental / Anti-Bacterial Agents / Entamoeba histolytica / Veterinary Sciences / Drug Targeting / Hydrogen-Ion Concentration / Disulfide bond

Lipids as clinical drugs, lipids as drug targets

Physical sciences / CHEMICAL SCIENCES / Estudents / Drug Targeting

Transient receptor potential (TRP) channels as drug targets

Transient receptor potential channels / Drug Design / Urinary Tract / Drug Targeting / Ligands

C. elegans: a novel pharmacogenetic model to study Parkinson\'s disease

Genetics / Cognitive Science / Caenorhabditis elegans / Molecular Mechanics / Protein-Protein Interaction / Tissue culture / Clinical Sciences / Dopamine Transporter / Model System / Degeneration / Genetic Analysis / Metabolic pathway / Drug Targeting / Substantia nigra pars compacta (SNpc) / Tissue culture / Clinical Sciences / Dopamine Transporter / Model System / Degeneration / Genetic Analysis / Metabolic pathway / Drug Targeting / Substantia nigra pars compacta (SNpc)

Myristoyl-CoA:Protein N-Myristoyltransferase, an Essential Enzyme and Potential Drug Target in Kinetoplastid Parasites

Kinetics / Drug development / Biological Chemistry / Leishmania / Cell Division / Biological Sciences / Saccharomyces cerevisiae / Molecular / RNA interference / Virulence / Cell line / Humans / Mice / Endocytosis / Animals / Cell Death / Biological / Polymerase Chain Reaction / Capsid / Phenotype / Enzyme / CHEMICAL SCIENCES / Mouse Model / Rats / Trypanosoma / Trypanosoma brucei / Time Factors / Trypanosoma brucei brucei / Isoenzymes / Fatty Acid / Protozoan Proteins / Species Specificity / Amino Acid Sequence / Subcellular Fractions / Golgi Apparatus / Recombinant Proteins / Drug Targeting / Cell Survival / Leishmania Major / Biochemistry and cell biology / Poliovirus / Immunoblotting / Biological Sciences / Saccharomyces cerevisiae / Molecular / RNA interference / Virulence / Cell line / Humans / Mice / Endocytosis / Animals / Cell Death / Biological / Polymerase Chain Reaction / Capsid / Phenotype / Enzyme / CHEMICAL SCIENCES / Mouse Model / Rats / Trypanosoma / Trypanosoma brucei / Time Factors / Trypanosoma brucei brucei / Isoenzymes / Fatty Acid / Protozoan Proteins / Species Specificity / Amino Acid Sequence / Subcellular Fractions / Golgi Apparatus / Recombinant Proteins / Drug Targeting / Cell Survival / Leishmania Major / Biochemistry and cell biology / Poliovirus / Immunoblotting

Myristoyl-CoA:protein N-myristoyltransferase, an essential enzyme and potential drug target in kinetoplastid parasites

Kinetics / Drug development / Biological Chemistry / Leishmania / Cell Division / Biological Sciences / Saccharomyces cerevisiae / Molecular / RNA interference / Virulence / Cell line / Humans / Mice / Endocytosis / Animals / Cell Death / Biological / Polymerase Chain Reaction / Capsid / Phenotype / Enzyme / CHEMICAL SCIENCES / Mouse Model / Rats / Trypanosoma / Trypanosoma brucei / Time Factors / Trypanosoma brucei brucei / Isoenzymes / Fatty Acid / Protozoan Proteins / Species Specificity / Amino Acid Sequence / Subcellular Fractions / Golgi Apparatus / Recombinant Proteins / Drug Targeting / Cell Survival / Leishmania Major / Biochemistry and cell biology / Poliovirus / Immunoblotting / Biological Sciences / Saccharomyces cerevisiae / Molecular / RNA interference / Virulence / Cell line / Humans / Mice / Endocytosis / Animals / Cell Death / Biological / Polymerase Chain Reaction / Capsid / Phenotype / Enzyme / CHEMICAL SCIENCES / Mouse Model / Rats / Trypanosoma / Trypanosoma brucei / Time Factors / Trypanosoma brucei brucei / Isoenzymes / Fatty Acid / Protozoan Proteins / Species Specificity / Amino Acid Sequence / Subcellular Fractions / Golgi Apparatus / Recombinant Proteins / Drug Targeting / Cell Survival / Leishmania Major / Biochemistry and cell biology / Poliovirus / Immunoblotting

LeishCyc: a biochemical pathways database for Leishmania major

Data Mining / Metabolomics / Proteomics / Humans / System Analysis / Animals / Error Correction / Genome Annotation / Spectrum / Digestive Tract / Plasmodium falciparum / Yeast Metabolite Profiling / Genome sequence / Protozoan Proteins / Metabolic pathway / Literature Search / Drug Targeting / Leishmania Major / Web Interface / Animals / Error Correction / Genome Annotation / Spectrum / Digestive Tract / Plasmodium falciparum / Yeast Metabolite Profiling / Genome sequence / Protozoan Proteins / Metabolic pathway / Literature Search / Drug Targeting / Leishmania Major / Web Interface

LeishCyc: a biochemical pathways database for Leishmania major

Data Mining / Metabolomics / Proteomics / Humans / System Analysis / Animals / Error Correction / Genome Annotation / Spectrum / Digestive Tract / Plasmodium falciparum / Yeast Metabolite Profiling / Genome sequence / Protozoan Proteins / Metabolic pathway / Literature Search / Drug Targeting / Leishmania Major / Web Interface / Animals / Error Correction / Genome Annotation / Spectrum / Digestive Tract / Plasmodium falciparum / Yeast Metabolite Profiling / Genome sequence / Protozoan Proteins / Metabolic pathway / Literature Search / Drug Targeting / Leishmania Major / Web Interface

Quinuclidine Derivatives as Potential Antiparasitics

Microbiology / Medical Microbiology / Animals / Enzyme / Rats / Trypanosoma Cruzi / Trypanosoma brucei / Trypanosoma brucei brucei / Plasmodium falciparum / Antimicrobial agents / Sterols / Structure activity Relationship / Recombinant Proteins / Drug Targeting / Leishmania Major / Plasma Membrane / Area of Interest / Molecular Structure / Trypanosoma Cruzi / Trypanosoma brucei / Trypanosoma brucei brucei / Plasmodium falciparum / Antimicrobial agents / Sterols / Structure activity Relationship / Recombinant Proteins / Drug Targeting / Leishmania Major / Plasma Membrane / Area of Interest / Molecular Structure

Targeting nucleotide dimers containing antiviral nucleosides

Drug delivery / Enzyme / Viral Infection / Combination drug therapy / Side Effect / Drug Targeting / Nucleotides / Drug Targeting / Nucleotides

Quinuclidine Derivatives as Potential Antiparasitics

Microbiology / Medical Microbiology / Animals / Enzyme / Rats / Trypanosoma Cruzi / Trypanosoma brucei / Trypanosoma brucei brucei / Plasmodium falciparum / Antimicrobial agents / Sterols / Structure activity Relationship / Recombinant Proteins / Drug Targeting / Leishmania Major / Plasma Membrane / Area of Interest / Molecular Structure / Trypanosoma Cruzi / Trypanosoma brucei / Trypanosoma brucei brucei / Plasmodium falciparum / Antimicrobial agents / Sterols / Structure activity Relationship / Recombinant Proteins / Drug Targeting / Leishmania Major / Plasma Membrane / Area of Interest / Molecular Structure

Lipids as clinical drugs, lipids as drug targets

Physical sciences / CHEMICAL SCIENCES / Estudents / Drug Targeting
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